SCHEMBL8554334

SCHEMBL8554334

COc1cc(OC(C)[C@@H]2CCCN2)cnc1F

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
KCNH2 Q12809 1/20 0.35
CHRNB4 P30926 4/20 0.34
CHRNA3 P32297 4/20 0.34
MAPK1 P28482 1/20 0.34
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551060 0.94 MEN1 (0.33) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8550718 0.94 MEN1 (0.33) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8622165 0.89 SLC6A2 (0.34) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8619125 0.89 SLC6A2 (0.34) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8556820 0.86 SLC6A2 (0.35) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8552875 0.85 SLC6A2 (0.33) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8551051 0.84 ADRA2A (0.33) SLC6A2SLC6A4
SCHEMBL8553260 0.80
SCHEMBL8551464 0.80
SCHEMBL8554797 0.79 IRAK4 (0.40) IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0846114-A1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1998-06-10 EP claimed
WO-1996040682-A1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1996-12-19 WO claimed
EP-0846114-A1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1998-06-10 EP disclosed
WO-1996040682-A1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1996-12-19 WO disclosed