SCHEMBL8554661

SCHEMBL8554661

O=[N+]([O-])c1ccc(CCN2CCNCCNCCNCC2)cc1

nearest known ligand 0.97

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 15/20 0.97
KCNH2 Q12809 14/20 0.97
HRH3 Q9Y5N1 1/20 0.72
SIGMAR1 Q99720 1/20 0.62
MAOA P21397 1/20 0.59
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
ADRB1 P08588 1/20 0.54
SIRT6 Q8N6T7 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9015442 1.00 KCNJ1 (0.97) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL2723268 0.98 KCNJ1 (1.00) KCNJ1KCNH2HRH3SIGMAR1MAOA
Hydrochloric Acid SCHEMBL286767 0.97 KCNJ1 (0.97) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL14478357 0.93 KCNJ1 (0.84) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL4549501 0.93 KCNJ1 (0.89) KCNJ1KCNH2HRH3SIGMAR1MAOA
Hydrochloric Acid SCHEMBL2731631 0.92 KCNJ1 (0.86) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL2731306 0.87 KCNJ1 (1.00) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL5334337 0.84 KCNJ1 (0.70) KCNJ1KCNH2HRH3SIGMAR1KDM4E
SCHEMBL5653299 0.84 HRH3 (0.93) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL3156895 0.84 HRH3 (1.00) KCNJ1KCNH2HRH3SIGMAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756065-A DIAGNOSTIC CHELATES FOR ANTIBODIES AND RADIOACTIVE MATERIALS THE DOW CHEMICAL COMPANY (US) 1998-05-26 US disclosed
EP-0374929-B1 Process for preparing mono-N-alkylated polyazamacrocycles DOW CHEMICAL CO (US) 1998-03-25 EP disclosed
US-5652361-A ANTITUMOR THE DOW CHEMICAL COMPANY (US) 1997-07-29 US disclosed
US-5435990-A Chelate-antibody complexes, treatment and diagnosis of cancer, tetraazacyclododecane compounds THE DOW CHEMICAL COMPANY (US) 1995-07-25 US disclosed
EP-0353450-B1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates DOW CHEMICAL CO (US) 1995-03-29 EP disclosed
US-5064956-A Process for preparing mono-n-alkylated polyazamacrocycles THE DOW CHEMICAL COMPANY (US) 1991-11-12 US disclosed
EP-0420942-A1 MACROCYCLIC BIFUNCTIONAL CHELANTS, COMPLEXES THEREOF AND THEIR ANTIBODY CONJUGATES THE DOW CHEMICAL COMPANY (US) 1991-04-10 EP disclosed
WO-1990007261-A2 PROCESS FOR PREPARING MONO-N-ALKYLATED POLYAZAMACROCYCLES THE DOW CHEMICAL COMPANY (US) 1990-07-12 WO disclosed
EP-0374929-A1 Process for preparing mono-n-alkylated polyazamacrocycles THE DOW CHEMICAL COMPANY (US) 1990-06-27 EP disclosed
EP-0353450-A1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates THE DOW CHEMICAL COMPANY (US) 1990-02-07 EP disclosed
WO-1989012631-A1 MACROCYCLIC BIFUNCTIONAL CHELANTS, COMPLEXES THEREOF AND THEIR ANTIBODY CONJUGATES THE DOW CHEMICAL COMPANY (US) 1989-12-28 WO disclosed