SCHEMBL8554737

SCHEMBL8554737

COc1ccc2c(c1)CCCN2N=O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.66
HSD17B10 Q99714 1/20 0.58
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
NOTUM Q6P988 1/20 0.51
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
TP53 P04637 1/20 0.47
DRD2 P14416 4/20 0.47
DRD1 P21728 4/20 0.47
DRD4 P21917 4/20 0.47
DRD5 P21918 4/20 0.47
DRD3 P35462 4/20 0.47
HDAC1 Q13547 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4102267 0.91 NOTUM (0.57) ALDH1A1HSD17B10KMT2AMEN1NOTUM
SCHEMBL2616321 0.78 HSD17B10 (0.60) ALDH1A1HSD17B10KMT2AMEN1NOTUM
SCHEMBL12061308 0.77 HRH3 (0.62) ALDH1A1HSD17B10KMT2AMEN1NOTUM
SCHEMBL7261315 0.76 HSD17B10 (0.62) HSD17B10KMT2AMEN1NOTUMPDK1
SCHEMBL7733872 0.76 ALDH1A1 (0.67) ALDH1A1NOTUMPDK1PDK2PDK3
SCHEMBL21524785 0.76 HSD17B10 (0.58) HSD17B10KMT2AMEN1NOTUMPDK1
SCHEMBL13531815 0.76 MEN1 (0.66) HSD17B10KMT2AMEN1NOTUMPDK1
SCHEMBL1177380 0.76 HSD17B10 (0.58) HSD17B10KMT2AMEN1NOTUMPDK1
SCHEMBL1177381 0.76 HSD17B10 (0.58) HSD17B10KMT2AMEN1NOTUMPDK1
SCHEMBL2203840 0.75 NOTUM (0.83) ALDH1A1HSD17B10KMT2AMEN1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529452-B1 1,7-Condensed 3-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SOLVAY PHARM GMBH (DE) 1998-11-11 EP disclosed
US-5324725-A Antiinflammatory agent, antiallergen KALI-CHEMIE PHARMA GMBH (DE) 1994-06-28 US disclosed
EP-0529452-A2 1,7-Condensed 2-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1993-03-03 EP disclosed