SCHEMBL8554934

SCHEMBL8554934

c1ccc(Cn2ccc3cc(Nc4ncnc5ccccc45)ccc32)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 10/20 1.00
EGFR P00533 9/20 0.68
ERBB4 Q15303 3/20 0.60
AURKB Q96GD4 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
CHEK2 O96017 1/20 0.52
ROS1 P08922 1/20 0.52
FLT3 P36888 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
DAPK3 O43293 1/20 0.51
MAP4K4 O95819 1/20 0.51
ABL1 P00519 1/20 0.51
PIM1 P11309 1/20 0.51
PRKACA P17612 1/20 0.51
LTK P29376 1/20 0.51
MAPK8 P45983 1/20 0.51
CSNK1A1 P48729 1/20 0.51
RPS6KA3 P51812 1/20 0.51
LIMK1 P53667 1/20 0.51
MAP2K1 Q02750 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31061496 1.00 ERBB2 (1.00) ERBB2EGFRERBB4AURKBCLK4
Hydrochloric Acid SCHEMBL8597573 0.99 ERBB2 (0.98) ERBB2EGFRERBB4AURKBCLK4
SCHEMBL9910675 0.89 EGFR (0.84) ERBB2EGFRERBB4
SCHEMBL6768642 0.86 ERBB2 (0.76) ERBB2EGFRERBB4MAP2K1
Hydrochloric Acid SCHEMBL6767640 0.86 ERBB2 (0.74) ERBB2EGFRERBB4MAP2K1
SCHEMBL8560522 0.85 ERBB2 (0.73) ERBB2EGFRERBB4ABL1
SCHEMBL8556847 0.85 ERBB2 (1.00) ERBB2EGFRERBB4ABCG2
Hydrochloric Acid SCHEMBL8596174 0.84 ERBB2 (0.98) ERBB2EGFRERBB4ABCG2
SCHEMBL8560791 0.84 ERBB2 (0.84) ERBB2EGFRERBB4
Hydrochloric Acid SCHEMBL8894449 0.84 ERBB2 (0.72) ERBB2EGFRERBB4ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-1975620-A2 Three hybrid assay system GPC Biotech AG (DE) 2008-10-01 EP disclosed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed