SCHEMBL8560522

SCHEMBL8560522

c1ccc(Cn2ccc3cc(Nc4ncnc5cc6c(cc45)OCO6)ccc32)cc1

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 7/20 0.73
EGFR P00533 11/20 0.61
ERBB4 Q15303 3/20 0.59
ABL1 P00519 3/20 0.58
PDGFRB P09619 3/20 0.58
FGFR1 P11362 3/20 0.58
SRC P12931 3/20 0.58
KDR P35968 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8894449 0.99 ERBB2 (0.72) ERBB2EGFRERBB4ABL1PDGFRB
SCHEMBL8554934 0.85 ERBB2 (1.00) ERBB2EGFRERBB4ABL1
SCHEMBL31061496 0.85 ERBB2 (1.00) ERBB2EGFRERBB4ABL1
Hydrochloric Acid SCHEMBL8597573 0.84 ERBB2 (0.98) ERBB2EGFRERBB4
SCHEMBL9910675 0.83 EGFR (0.84) ERBB2EGFRERBB4
SCHEMBL8556847 0.83 ERBB2 (1.00) ERBB2EGFRERBB4KDR
SCHEMBL6768642 0.82 ERBB2 (0.76) ERBB2EGFRERBB4
SCHEMBL8560791 0.82 ERBB2 (0.84) ERBB2EGFRERBB4KDR
Hydrochloric Acid SCHEMBL8596174 0.82 ERBB2 (0.98) ERBB2EGFRERBB4KDR
Hydrochloric Acid SCHEMBL6767640 0.82 ERBB2 (0.74) ERBB2EGFRERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed