SCHEMBL8554985

SCHEMBL8554985

O=C1[N]c2c(cc(Cl)c([N+](=O)[O-])c2Cl)NC1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
TSHR P16473 2/20 0.40
GRIN2D O15399 10/20 0.36
GRIN3B O60391 10/20 0.36
GRIN1 Q05586 10/20 0.36
GRIN2A Q12879 10/20 0.36
GRIN2B Q13224 10/20 0.36
GRIN2C Q14957 10/20 0.36
GRIN3A Q8TCU5 10/20 0.36
CES1 P23141 1/20 0.33
CAPN9 O14815 1/20 0.32
CASP3 P42574 1/20 0.32
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
XBP1 P17861 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5274587 0.88 TSHR (0.47) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8556823 0.86 GRIN2D (0.35) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8558654 0.86 TSHR (0.38) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8113141 0.83 GRIN2D (0.45) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8114652 0.83 TSHR (0.34) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8554603 0.82 TSHR (0.34) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8122907 0.81 TSHR (0.35) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL7352737 0.80 TSHR (0.34) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8121622 0.80 GRIN2D (0.45) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL8113964 0.80 GRIN2D (0.38) ALDH1A1TSHRGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed