SCHEMBL8555480

SCHEMBL8555480

CC(C(N)=O)(c1ccccc1)N1C(=O)C(NC(=O)O)N=C(CBr)c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 13/20 0.38
SCN9A Q15858 1/20 0.36
NOTCH1 P46531 2/20 0.35
NOTCH3 Q9UM47 1/20 0.35
CCKAR P32238 4/20 0.35
KCNH2 Q12809 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
RBPJ Q06330 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927644 0.60 CCKBR (0.78) CCKBRCCKAR
SCHEMBL7207460 0.60 CCKBR (0.78) CCKBRCCKAR
SCHEMBL9272046 0.56 CYP11B1 (0.54) CCKBRKCNH2
SCHEMBL5706512 0.56 KMT2A (0.44)
SCHEMBL7746365 0.56 MAPT (0.39)
SCHEMBL11602590 0.54 MAPT (0.65) KCNH2
Atrolactamide SCHEMBL78236 0.54 MAPT (0.65) KCNH2
Ethane SCHEMBL3002447 0.54 MAPT (0.59) KCNH2
SCHEMBL6266546 0.54 CYP2B6 (0.56)
SCHEMBL14477084 0.54 CA12 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672037-B1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LTD (GB) 1998-07-08 EP disclosed