SCHEMBL8555578

SCHEMBL8555578

C=C1N(CCCCCCCCCCCC)c2ccccc2C1(C)C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CES1 P23141 2/20 0.46
CDC25A P30304 1/20 0.46
SCN9A Q15858 7/20 0.45
ALDH1A1 P00352 3/20 0.43
ALDH2 P05091 1/20 0.43
ALDH3A1 P30838 1/20 0.43
CNR2 P34972 2/20 0.42
MEN1 O00255 2/20 0.41
GLA P06280 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14134758 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL9868831 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL8708894 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL9736812 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL8475420 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL19746373 1.00 KMT2A (0.50) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL10448669 0.98 KMT2A (0.51) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL6093583 0.94 KMT2A (0.53) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL30996203 0.94 CYP1A2 (0.55) KMT2ACYP1A2CYP2D6CES1CDC25A
SCHEMBL30996195 0.88 KMT2A (0.40) KMT2ACYP1A2CYP2D6CES1CDC25A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529100-B1 INDOLINOSPIROBENZOPYRAN DERIVATIVE OTSUKA KAGAKU KK (JP) 1998-11-11 EP disclosed
EP-0530369-B1 CRYSTAL COMPRISING INDOLINOSPIROBENZOTHIOPYRAN DERIVATIVE AND RING-OPENING ISOMER THEREOF OTSUKA KAGAKU KK (JP) 1997-02-05 EP disclosed
US-5403702-A Crystals consisting of an indolinospirobenzopyran derivative OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1995-04-04 US disclosed
US-5320784-A Crystal comprising an indolinospirobenzothiopyran derivative and its ring opened isomer OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1994-06-14 US disclosed
EP-0530369-A1 CRYSTAL COMPRISING INDOLINOSPIROBENZOTHIOPYRAN DERIVATIVE AND RING-OPENING ISOMER THEREOF OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1993-03-10 EP disclosed
EP-0529100-A1 INDOLINOSPIROBENZOPYRAN DERIVATIVE OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1993-03-03 EP disclosed