SCHEMBL8555902

SCHEMBL8555902

CC(C)(C)OC(=O)NC1CCc2[nH]c3ccc(OCc4ccccc4)cc3c2C1.CNC1CCc2[nH]c3ccc(O)cc3c2C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
HTR1B P28222 2/20 0.47
HTR1D P28221 1/20 0.47
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
HTR1E P28566 1/20 0.47
HTR7 P34969 1/20 0.47
OPRM1 P35372 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
MAPKAPK2 P49137 1/20 0.44
EGFR P00533 1/20 0.44
IGF1R P08069 1/20 0.44
FLT4 P35916 1/20 0.44
KDR P35968 1/20 0.44
S1PR1 P21453 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7663983 0.94 MAPKAPK2 (0.49) HTR1AHTR1BHTR1DDRD2DRD4
SCHEMBL8608335 0.87 MAPKAPK2 (0.42) HTR1BHTR1DMAPKAPK2EGFRIGF1R
SCHEMBL7662787 0.86 HTR1B (0.53) HTR1AHTR1BHTR1DDRD2DRD4
SCHEMBL8559020 0.82 EGFR (0.50) HTR1BHTR1DMAPKAPK2EGFRIGF1R
SCHEMBL24408396 0.79 HTR1B (0.57) HTR1AHTR1BHTR1DDRD2DRD4
SCHEMBL7655639 0.77 HTR1D (0.50) HTR1BHTR1DMAPKAPK2EGFRIGF1R
SCHEMBL11418263 0.76 MCHR1 (0.49)
SCHEMBL834332 0.76 MEN1 (0.53) HTR1AHTR1BHTR1D
SCHEMBL1905530 0.76 MEN1 (0.53) HTR1AHTR1BHTR1D
SCHEMBL834331 0.76 MEN1 (0.53) HTR1AHTR1BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708187-A MIGRANE HEADACHES ELI LILLY AND COMPANY (US) 1998-01-13 US disclosed