SCHEMBL8556917

SCHEMBL8556917

Cc1cc(C(=O)N2Cc3ccccc3Cc3ccccc32)ccc1[N+](=O)[O-]

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
BLM P54132 1/20 0.49
GAA P10253 4/20 0.48
MAPT P10636 3/20 0.48
MGAM O43451 1/20 0.48
AMY1A P0DUB6 1/20 0.48
SI P14410 1/20 0.48
MGAM2 Q2M2H8 1/20 0.48
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
NPBWR1 P48145 1/20 0.47
MCHR1 Q99705 1/20 0.47
POLB P06746 1/20 0.46
AVPR2 P30518 1/20 0.45
AVPR1A P37288 1/20 0.45
HSP90AA1 P07900 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349544 0.82 KMT2A (0.53) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL7331322 0.82 AVPR1A (0.69) AVPR2AVPR1A
SCHEMBL8556540 0.81 HSD17B3 (0.45) MEN1KMT2ASMN1; SMN2AVPR2AVPR1A
SCHEMBL7346893 0.81 MEN1 (0.68) ALDH1A1MEN1KMT2AMAPTAVPR2
SCHEMBL7360343 0.77 AVPR1A (0.44) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL7340153 0.76 AVPR1A (0.43) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL8560249 0.73 HPGD (0.53) ALDH1A1KMT2ATSHRSMN1; SMN2AVPR2
SCHEMBL8558207 0.72 AVPR2 (0.60) ALDH1A1KMT2ASMN1; SMN2AVPR2AVPR1A
SCHEMBL8558342 0.72 HPGD (0.48) ALDH1A1KMT2ASMN1; SMN2AVPR2AVPR1A
SCHEMBL8559036 0.72 HPGD (0.50) ALDH1A1MEN1KMT2AL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed