SCHEMBL8557426

SCHEMBL8557426

O=C(Nc1ccc(C(=O)N2Cc3ccccc3Oc3ccccc32)cc1)c1cccc(Cl)c1Cl

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
AVPR2 P30518 3/20 0.48
AVPR1A P37288 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561438 0.85 AVPR2 (0.59) AVPR2AVPR1A
SCHEMBL7340029 0.85 AVPR2 (0.50) AVPR2AVPR1A
SCHEMBL8562440 0.85 AVPR2 (0.54) AVPR2AVPR1A
SCHEMBL8559574 0.85 AVPR1A (0.56) AVPR2AVPR1A
SCHEMBL7337255 0.83 AVPR2 (0.63) AVPR2AVPR1A
SCHEMBL8556495 0.83 AVPR2 (0.55) AVPR2AVPR1A
SCHEMBL8565042 0.81 AVPR2 (0.62) NPC1RAB9AAVPR2AVPR1A
SCHEMBL8563252 0.80 TP53 (0.47)
SCHEMBL8563988 0.80 AVPR1A (0.58) AVPR2AVPR1A
SCHEMBL8561578 0.79 AVPR1A (0.55) NPC1RAB9AAVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed