SCHEMBL8557797

SCHEMBL8557797

CS(=O)(=O)[N+]1(NC(=O)C(COCc2ccccc2)NC(=O)c2cccc3ccccc23)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.35
CTSS P25774 2/20 0.35
CTSV O60911 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
GHSR Q92847 1/20 0.34
KCNA5 P22460 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561114 0.90 TACR1 (0.40) TACR1GHSR
SCHEMBL8559324 0.90 KCNA5 (0.38) TACR1CTSSCTSLKCNA5
SCHEMBL8559848 0.89 TACR1 (0.40) TACR1
Hydrochloric Acid SCHEMBL8563552 0.89 KCNA5 (0.38) TACR1CTSSCTSLKCNA5
SCHEMBL8561651 0.89 TACR1 (0.42) TACR1GHSR
SCHEMBL8563529 0.87 TACR1 (0.41) TACR1
SCHEMBL8559389 0.87 TACR1 (0.42) TACR1CTSSCTSLGHSR
SCHEMBL8559555 0.87 TACR1 (0.40) TACR1GHSR
SCHEMBL8559045 0.86 TACR1 (0.41) TACR1CTSB
SCHEMBL8560138 0.86 TACR1 (0.41) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed