SCHEMBL8558035

SCHEMBL8558035

CC1=NC(NC(=O)Nc2cccc(C)c2)C(=O)Nc2c(C)cccc21

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 17/20 0.62
KCNH2 Q12809 1/20 0.48
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550799 0.86 CCKBR (0.78) CCKBRKCNH2MAPT
SCHEMBL7550802 0.86 CCKBR (0.78) CCKBRKCNH2MAPT
SCHEMBL7546371 0.78 CCKBR (0.65) CCKBRKCNH2
SCHEMBL641958 0.76 CCKBR (1.00) CCKBRKCNH2CYP3A4MAPTTSHR
SCHEMBL7547182 0.76 CCKBR (0.72) CCKBRKCNH2MAPT
SCHEMBL7547190 0.76 CCKBR (0.72) CCKBRKCNH2MAPT
SCHEMBL7552167 0.76 CCKBR (0.75) CCKBRKCNH2MAPT
SCHEMBL7552157 0.76 CCKBR (0.75) CCKBRKCNH2MAPT
SCHEMBL9866481 0.76 CCKBR (0.64) CCKBRKCNH2
SCHEMBL7545616 0.75 CYP3A4 (0.60) CCKBRCYP3A4MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934282-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
WO-1998015535-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-16 WO disclosed