SCHEMBL8558265

SCHEMBL8558265

c1ccc(Cn2cnc3cc(Nc4ncnc5ccccc45)ccc32)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 7/20 1.00
NR1I2 O75469 7/20 0.53
EGFR P00533 4/20 0.53
AURKB Q96GD4 2/20 0.53
CLK4 Q9HAZ1 2/20 0.53
CHEK2 O96017 1/20 0.53
ROS1 P08922 1/20 0.53
FLT3 P36888 1/20 0.53
ERBB4 Q15303 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
TNF P01375 1/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
DAPK3 O43293 1/20 0.52
MAP4K4 O95819 1/20 0.52
ABL1 P00519 1/20 0.52
PIM1 P11309 1/20 0.52
PRKACA P17612 1/20 0.52
LTK P29376 1/20 0.52
MAPK8 P45983 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8893805 0.99 ERBB2 (0.98) ERBB2NR1I2EGFRAURKBCLK4
SCHEMBL8560275 0.91 ERBB2 (1.00) ERBB2NR1I2EGFRAURKBCLK4
Hydrochloric Acid SCHEMBL8895524 0.90 ERBB2 (0.98) ERBB2NR1I2EGFRAURKBCLK4
SCHEMBL8554934 0.83 ERBB2 (1.00) ERBB2EGFRAURKBCLK4CHEK2
SCHEMBL31061496 0.83 ERBB2 (1.00) ERBB2EGFRAURKBCLK4CHEK2
Hydrochloric Acid SCHEMBL8597573 0.82 ERBB2 (0.98) ERBB2EGFRAURKBCLK4CHEK2
SCHEMBL31061501 0.78 ERBB2 (0.76) ERBB2EGFRERBB4MAP2K1
SCHEMBL8561085 0.78 ERBB2 (0.76) ERBB2EGFRERBB4MAP2K1
Hydrochloric Acid SCHEMBL8557183 0.74 ERBB2 (0.59) ERBB2NR1I2TNFCYP11B1CYP11B2
SCHEMBL7119433 0.74 ERBB2 (0.68) ERBB2EGFRERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed