SCHEMBL8558469

SCHEMBL8558469

c1ccc(Cc2nc3cc(Nc4ncnc5ccccc45)ccc3[nH]2)cc1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 9/20 0.85
KDR P35968 6/20 0.56
MET P08581 5/20 0.56
EGFR P00533 4/20 0.53
AURKB Q96GD4 2/20 0.53
CLK4 Q9HAZ1 2/20 0.53
CHEK2 O96017 1/20 0.53
ROS1 P08922 1/20 0.53
FLT3 P36888 1/20 0.53
ERBB4 Q15303 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
GAA P10253 1/20 0.52
DAPK3 O43293 1/20 0.52
MAP4K4 O95819 1/20 0.52
ABL1 P00519 1/20 0.52
PIM1 P11309 1/20 0.52
PRKACA P17612 1/20 0.52
LTK P29376 1/20 0.52
MAPK8 P45983 1/20 0.52
CSNK1A1 P48729 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8893639 0.99 ERBB2 (0.84) ERBB2KDRMETEGFRAURKB
SCHEMBL8558474 0.92 ERBB2 (1.00) ERBB2KDRMETEGFR
Hydrochloric Acid SCHEMBL8893650 0.91 ERBB2 (0.98) ERBB2KDRMETEGFR
SCHEMBL4354490 0.85 ERBB2 (0.68) ERBB2KDRMETEGFRERBB4
SCHEMBL8555750 0.84 ERBB2 (0.87) ERBB2KDREGFRABCG2
Hydrochloric Acid SCHEMBL8894692 0.84 ERBB2 (0.86) ERBB2KDREGFRABCG2
Gw301888X SCHEMBL6765469 0.83 ERBB2 (0.65) ERBB2EGFRERBB4MAP2K1
SCHEMBL7126243 0.83 EGFR (0.62) ERBB2EGFRERBB4
SCHEMBL7119435 0.82 FYN (0.66) ERBB2EGFRERBB4
SCHEMBL5922764 0.80 ERBB2 (0.57) ERBB2KDREGFRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-1364212-B1 THREE HYBRID ASSAY SYSTEM GPC BIOTECH AG (DE) 2011-02-02 EP disclosed
EP-1975620-A2 Three hybrid assay system GPC Biotech AG (DE) 2008-10-01 EP disclosed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed