SCHEMBL8559064

SCHEMBL8559064

Clc1cccc2c1Sc1ccccc1NC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.41
HSD17B10 Q99714 1/20 0.41
GAA P10253 6/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MAPT P10636 6/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALOX12 P18054 2/20 0.37
BCHE P06276 2/20 0.37
ACHE P22303 2/20 0.37
NOX1 Q9Y5S8 2/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
MAOA P21397 1/20 0.37
CNR1 P21554 1/20 0.37
PTGS1 P23219 1/20 0.37
SLC6A2 P23975 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558840 0.83 NOX1 (0.43) ALOX15HSD17B10GAANPSR1MAPT
SCHEMBL8561569 0.81 MEN1 (0.47) ALOX15HSD17B10GAANPSR1MAPT
SCHEMBL4510651 0.77 GAA (0.52) ALOX15HSD17B10GAANPSR1MAPT
SCHEMBL7069691 0.74 NOX1 (0.59) ALOX15GAANPSR1MAPTMEN1
SCHEMBL8817021 0.74 MEN1 (0.45) NPSR1MAPTMEN1KMT2AALOX12
SCHEMBL8558177 0.71 NOX1 (0.58) ALOX15HSD17B10GAANPSR1MAPT
SCHEMBL25002667 0.69 MEN1 (0.48) NPSR1MAPTMEN1KMT2AALOX12
SCHEMBL8559836 0.69 MEN1 (0.36) GAANPSR1MAPTMEN1KMT2A
SCHEMBL8556950 0.69 NOX1 (0.41) GAAMAPTMEN1KMT2ABCHE
SCHEMBL8562468 0.68 NOX1 (0.58) ALOX15HSD17B10GAANPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed