SCHEMBL8559657

SCHEMBL8559657

CCC(C)OC(=O)C1C=Cc2ccccc2N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
P2RX4 Q99571 2/20 0.34
ADORA2B P29275 2/20 0.34
GABRA1 P14867 3/20 0.33
GABRG2 P18507 3/20 0.33
GABRB3 P28472 3/20 0.33
GABRA5 P31644 3/20 0.33
GABRA3 P34903 3/20 0.33
GABRA2 P47869 3/20 0.33
GABRA6 Q16445 1/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 1/20 0.32
ADRA1A P35348 1/20 0.31
KDM4E B2RXH2 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11386324 0.86 P2RX4 (0.37) MAPTP2RX4TSHRSMN1; SMN2LMNA
SCHEMBL4698118 0.81 KDM4E (0.43) MAPTCYP1A2TSHRCYP2C19SMN1; SMN2
SCHEMBL3250625 0.79 MAPT (0.40) MAPTP2RX4HSD17B10TSHRSMN1; SMN2
SCHEMBL14921032 0.75 EPHX2 (0.36) MAPTP2RX4SMN1; SMN2LMNAGAA
SCHEMBL30805659 0.75 EPHX2 (0.36) MAPTP2RX4SMN1; SMN2LMNAGAA
SCHEMBL28219643 0.73 FABP7 (0.43) P2RX4TSHRLMNAALDH1A1
SCHEMBL385982 0.72 MAPT (0.40) MAPTP2RX4HSD17B10CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL7435031 0.70 MAPT (0.39) MAPTP2RX4HSD17B10CYP3A4CYP2C9
SCHEMBL1286805 0.70 MAPT (0.38) MAPTP2RX4TSHRSMN1; SMN2LMNA
SCHEMBL31301236 0.70 MAPT (0.38) MAPTP2RX4TSHRSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756739-A Process for preparing polyamine derivative and intermediates thereof MERRELL PHARMACEUTICALS INC. (US) 1998-05-26 US disclosed
US-4207322-A 6-Aryl-s-triazolo-(4,3-alpha)-pyrido-(2,3-f)-(1,4)-diazepines DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1980-06-10 US disclosed
US-4110455-A 6-ARYL-S-TRIAZOLO-(4,3-A)-PYRIDO-(2,3-F)-1,4-DIAZEPINES DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1978-08-29 US disclosed