SCHEMBL8559837

SCHEMBL8559837

NC(=O)OC1NCCc2cc(O)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
KDM1A O60341 5/20 0.42
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
BCHE P06276 1/20 0.38
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
MAOA P21397 1/20 0.36
SLC6A9 P48067 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
DRD3 P35462 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560578 0.88 DRD2 (0.42) CA1CA2CA7CA9CA14
SCHEMBL27498312 0.87 HTR2A (0.44) CA1CA2CA7CA9CA14
Hydrochloric Acid SCHEMBL1022841 0.83 CA1 (0.43) CA1CA2CA7CA9CA14
SCHEMBL5161528 0.80 TSHR (0.54) TSHR
SCHEMBL27527951 0.78 HTR2A (0.46) KDM1AADRB1SLC6A9
SCHEMBL4573507 0.74 TSHR (0.62) CA1CA2CA7CA9CA14
SCHEMBL14267384 0.73 CA1 (0.51) CA1CA2CA7CA9CA14
SCHEMBL7124159 0.72 CA1 (0.46) CA1CA2CA7CA9CA14
SCHEMBL7199949 0.71 CA1 (0.52) CA1CA2CA7CA9CA14
Hydrochloric Acid SCHEMBL3534709 0.71 CA1 (0.45) CA1CA2CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1240448-A Method of preparation of physostigmine carbamate derivatives from eseproline ethers HOECHST MARION ROUSSEL INC (US) 2000-01-05 CN claimed
CN-1235607-A Preparation of physostigmine carbamate derivatives from eseretholes HOECHST MARION ROUSSEL INC (US) 1999-11-17 CN claimed
CN-1240448-A Method of preparation of physostigmine carbamate derivatives from eseproline ethers HOECHST MARION ROUSSEL INC (US) 2000-01-05 CN disclosed
CN-1235607-A Preparation of physostigmine carbamate derivatives from eseretholes HOECHST MARION ROUSSEL INC (US) 1999-11-17 CN disclosed
EP-0538248-B1 TETRAHYDROISOQUINOLINYLCARBAMATES OF 1,2,3,3A,8,8A-HEXAHYDRO-1,3A,8-TRIMETHYLPYRROLO [2,3-B]INDOLE HOECHST MARION ROUSSEL INC (US) 1998-02-11 EP disclosed