SCHEMBL8559895

SCHEMBL8559895

Cc1ccc(S(=O)(=O)OC(=O)[C@@H](N)CN)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
F2 P00734 3/20 0.40
PRSS1 P07477 3/20 0.40
PRSS2 P07478 3/20 0.40
PRSS3 P35030 3/20 0.40
GBA1 P04062 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 2/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9091962 1.00 ALDH1A1 (0.50) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL12572597 0.88 ALDH1A1 (0.47) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL28674512 0.88 ALDH1A1 (0.50) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL27692485 0.88 ALDH1A1 (0.50) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL28510750 0.88 ALDH1A1 (0.50) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL10378708 0.86 ALDH1A1 (0.49) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL9592709 0.85 ALDH1A1 (0.47) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL16464668 0.85 ALDH1A1 (0.47) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL28693501 0.85 ALDH1A1 (0.47) ALDH1A1F2PRSS1PRSS2PRSS3
SCHEMBL28583480 0.84 ALDH1A1 (0.44) ALDH1A1F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP disclosed
WO-1996038426-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-05 WO disclosed