SCHEMBL8560232

SCHEMBL8560232

O=C(Nc1cccc2[nH]cnc12)c1c(Cl)cccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 5/20 0.52
JAK2 O60674 4/20 0.52
JAK1 P23458 3/20 0.52
HDAC3 O15379 1/20 0.48
BRD4 O60885 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
PTGES O14684 2/20 0.46
RXFP1 Q9HBX9 1/20 0.46
CYP3A4 P08684 1/20 0.46
PARP1 P09874 1/20 0.46
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8473992 0.78 PARP1 (0.51) TYK2JAK2JAK1PTGESPARP1
SCHEMBL13135977 0.78 PARP1 (0.51) HDAC3BRD4HDAC4HDAC1HDAC7
SCHEMBL27660069 0.78 PARP1 (0.59) HDAC3BRD4HDAC4HDAC1HDAC7
SCHEMBL27888402 0.78 PARP1 (0.59) HDAC3BRD4HDAC4HDAC1HDAC7
SCHEMBL24534325 0.77 HDAC3 (0.50) HDAC3BRD4HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL28155445 0.77 PARP1 (0.58) HDAC3BRD4HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL27660077 0.77 PARP1 (0.58) HDAC3BRD4HDAC4HDAC1HDAC7
SCHEMBL196738 0.77 PARP1 (0.56) JAK2BRD4PARP1MEN1KMT2A
SCHEMBL8569632 0.76 TRPV1 (0.58) TYK2JAK2JAK1PTGESCYP3A4
SCHEMBL8597761 0.76 PTGES (0.52) TYK2JAK2JAK1PTGESMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed