Bromide

Bromide

SCHEMBL8560844

Br.O=C1c2ccccc2C(=O)c2c(CC3CCCCN3)cccc21

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
HTR6 P50406 10/20 0.42
KMT2A Q03164 1/20 0.41
MAPT P10636 2/20 0.40
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTR2A P28223 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP3A5 P20815 2/20 0.39
CYP3A7 P24462 2/20 0.39
CYP2C19 P33261 2/20 0.39
PDK4 Q16654 2/20 0.39
CYP3A43 Q9HB55 2/20 0.39
ALDH1A1 P00352 1/20 0.38
EGFR P00533 1/20 0.38
RAF1 P04049 1/20 0.38
ALOX12 P18054 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7739261 0.73 MAPT (0.39) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL7738544 0.72 MAPT (0.40) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL7737740 0.72 MAPT (0.40) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL7737941 0.72 MAPT (0.40) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL7738515 0.72 MAPT (0.40) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL11358872 0.72 CYP2D6 (0.59) POLBHTR6HTR2ACYP1A2CYP3A4
SCHEMBL7739394 0.71 MAPT (0.40) KMT2AMAPTMAPK1LMNAHPGD
SCHEMBL20828122 0.71 POLB (0.60) POLBHTR6KMT2AHTR2AHRH3
SCHEMBL17979696 0.71 POLB (0.60) POLBHTR6KMT2AHTR2AHRH3
SCHEMBL478235 0.71 POLB (0.60) POLBHTR6KMT2AHTR2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817842-A Process for the preparation of epoxides from olefins ENICHEM S.P.A. (IT) 1998-10-06 US disclosed
EP-0819683-A1 Process for the preparation of epoxides from olefins ENICHEM S.p.A. (IT) 1998-01-21 EP disclosed