SCHEMBL8563060

SCHEMBL8563060

COC(=O)c1ccc(CCN2CCN(c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)C2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.45
ESR1 P03372 3/20 0.41
ESR2 Q92731 3/20 0.41
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
S1PR1 P21453 1/20 0.38
HDAC6 Q9UBN7 1/20 0.37
DRD2 P14416 4/20 0.36
DRD3 P35462 4/20 0.36
KCNH2 Q12809 4/20 0.36
MAPT P10636 1/20 0.35
ABCB1 P08183 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
P2RX3 P56373 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566035 0.81 ESR1 (0.40) ESR1ESR2HDAC6ABCB1ABCG2
SCHEMBL7474127 0.79 TMEM97 (0.43) ESR1ESR2S1PR1DRD2DRD3
Hydrochloric Acid SCHEMBL8558787 0.78 HDAC1 (0.52) HDAC1GRIN1GRIN2BS1PR1DRD2
SCHEMBL7560796 0.77 ESR1 (0.42) ESR1ESR2HDAC6DRD2DRD3
SCHEMBL7283756 0.75 HDAC1 (0.55) HDAC1S1PR1
SCHEMBL8565997 0.74 ESR1 (0.40) ESR1ESR2HDAC6MAPT
SCHEMBL7281726 0.74 HDAC1 (0.54) HDAC1S1PR1HDAC6KCNH2
Hydrochloric Acid SCHEMBL8561009 0.72 HDAC1 (0.50) HDAC1GRIN1GRIN2BS1PR1
SCHEMBL8567198 0.72 ESR1 (0.43) HDAC1ESR1ESR2HDAC6MAPT
SCHEMBL8567193 0.72 ESR1 (0.43) HDAC1ESR1ESR2HDAC6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed