SCHEMBL8565997

SCHEMBL8565997

CCN1CC(c2ccc(C(=O)OC)cc2)N(c2ccc3c(c2)CCN(C(=O)C(F)(F)F)CC3)C1=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
HDAC6 Q9UBN7 2/20 0.39
HDAC8 Q9BY41 1/20 0.34
XIAP P98170 1/20 0.34
BIRC2 Q13490 1/20 0.34
TP53 P04637 3/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 2/20 0.34
TSHR P16473 1/20 0.34
GRM2 Q14416 1/20 0.33
MCHR1 Q99705 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
LMNA P02545 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563060 0.74 HDAC1 (0.45) ESR1ESR2HDAC6MAPT
SCHEMBL8561721 0.72 ESR1 (0.40) ESR1ESR2HDAC6HDAC8TP53
SCHEMBL8565993 0.71 ESR1 (0.40) ESR1ESR2HDAC6HDAC8TP53
SCHEMBL8566035 0.70 ESR1 (0.40) ESR1ESR2HDAC6SMN1; SMN2
SCHEMBL8558363 0.69 ESR1 (0.38) ESR1ESR2HDAC6SMN1; SMN2PDE4B
SCHEMBL8283285 0.69 ESR2 (0.70) ESR1ESR2HDAC6HDAC8MAPK1
SCHEMBL5359582 0.69 ESR1 (0.65) ESR1ESR2HDAC6HDAC8MAPK1
SCHEMBL7560796 0.69 ESR1 (0.42) ESR1ESR2HDAC6MAPTTSHR
SCHEMBL8563251 0.68 ESR1 (0.39) ESR1ESR2HDAC6SMN1; SMN2PDE4B
SCHEMBL14334874 0.67 ESR1 (0.45) ESR1ESR2HDAC6GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed