SCHEMBL8564001

SCHEMBL8564001

Clc1cc(Cl)c2nc(-c3cccc4ccccc34)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.57
ADORA3 P0DMS8 1/20 0.53
ADORA1 P30542 1/20 0.53
GAA P10253 2/20 0.49
MGAM O43451 1/20 0.49
SI P14410 1/20 0.49
MGAM2 Q2M2H8 1/20 0.49
PTGES O14684 5/20 0.48
HTT P42858 1/20 0.46
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
DHODH Q02127 3/20 0.44
PARP1 P09874 1/20 0.44
RHEB Q15382 1/20 0.41
GUSB P08236 1/20 0.40
MEN1 O00255 1/20 0.40
MITF O75030 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2951540 0.78 ALDH1A1 (0.61) CBFBADORA3KDM4EALDH1A1NPC1
SCHEMBL22955432 0.77 NPC1 (0.61) CBFBKDM4EALDH1A1NPC1RAB9A
SCHEMBL29824605 0.75 NPC1 (0.49) CBFBGAAPTGESHTTKDM4E
SCHEMBL2951537 0.75 NPC1 (0.49) CBFBGAAPTGESHTTKDM4E
SCHEMBL17829671 0.72 GUSB (0.58) PTGESPARP1GUSBTYMPPIM1
SCHEMBL124230 0.72 CBFB (1.00) CBFBADORA3ADORA1KDM4EALDH1A1
SCHEMBL1133803 0.72 NPC1 (0.52) GAAMGAMSIMGAM2PTGES
SCHEMBL5201397 0.72 MGAM (0.68) CBFBADORA3ADORA1GAAMGAM
SCHEMBL784353 0.70 NPC1 (0.66) GAAHTTKDM4EALDH1A1NPC1
SCHEMBL29825055 0.70 NPC1 (0.66) GAAHTTKDM4EALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed