SCHEMBL8564509

SCHEMBL8564509

C#CCC(=O)c1ccc(C(=O)OC(C)(C)C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.49
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
CA14 Q9ULX7 2/20 0.47
GABRA1 P14867 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
SLC7A5 Q01650 1/20 0.38
STAT3 P40763 2/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 2/20 0.37
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109451 0.82 CA1 (0.61) ELANECA12CA1CA2CA9
SCHEMBL8563045 0.81 CA12 (0.50) ELANECA12CA1CA2CA9
SCHEMBL925696 0.81 CA1 (0.53) CA12CA1CA2CA9CA14
SCHEMBL433863 0.80 ELANE (0.44) ELANECA12CA1CA2CA9
SCHEMBL24812731 0.80 GSK3B (0.55) ELANECA12CA1CA2CA9
SCHEMBL6258711 0.80 GABRA1 (0.50) ELANECA12CA1CA2CA9
Hydrazine SCHEMBL10771056 0.78 CA12 (0.62) ELANECA12CA1CA2CA9
SCHEMBL14661860 0.77 CA12 (0.46) ELANECA12CA1CA2CA9
SCHEMBL27960488 0.77 CA12 (0.46) ELANECA12CA1CA2CA9
SCHEMBL7196365 0.77 CA12 (0.53) ELANECA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed