SCHEMBL8564545

SCHEMBL8564545

CC(C)(C)OC(=O)c1ccc(CCCBr)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.45
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
PRNP P04156 1/20 0.41
RECQL P46063 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPSR1 Q6W5P4 2/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HDAC6 Q9UBN7 3/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC3 O15379 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
PRSS1 P07477 4/20 0.32
TMPRSS15 P98073 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4179468 0.88 HPGD (0.40) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8570240 0.87 HPGD (0.43) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL21199747 0.85 POLB (0.46) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8982459 0.85 HPGD (0.45) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL5050275 0.85 HPGD (0.42) HPGDALDH1A1LMNAPRNPRECQL
Hydrochloric Acid SCHEMBL5724631 0.84 HPGD (0.41) HPGDALDH1A1LMNAPRNPRECQL
Hydrochloric Acid SCHEMBL2413233 0.84 HPGD (0.40) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL9439542 0.83 HPGD (0.67) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL317871 0.83 HPGD (0.55) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8982537 0.83 HPGD (0.40) HPGDALDH1A1LMNAPRNPRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed