SCHEMBL8565103

SCHEMBL8565103

Cn1nc(-c2cc(N)c(F)cc2F)c(Cl)c1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
BRD4 O60885 1/20 0.35
HSD11B1 P28845 2/20 0.30
SLC34A1 Q06495 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
POLB P06746 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6289041 0.90 MEN1 (0.36) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8566222 0.85 MEN1 (0.38) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8566825 0.83 GAA (0.36) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8570221 0.80 MEN1 (0.37) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL7524976 0.80 CYP1A2 (0.39) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL7894519 0.80 NOTUM (0.32) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8564686 0.79 MEN1 (0.36) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL27322874 0.79 MEN1 (0.36) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL7615238 0.79 MEN1 (0.36) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8569766 0.78 HSD11B1 (0.47) MEN1CYP1A2CYP2C9CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1050121-C Process for preparing substituted aryl-halogenoalkyl pyrazoles MONSANTO CO (US) 2000-03-08 CN disclosed
EP-0553307-B1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO CO (US) 1998-12-09 EP disclosed
EP-0791571-A1 Benzoyl derivatives MONSANTO COMPANY (US) 1997-08-27 EP disclosed
US-5536700-A Herbicidal compositions comprising aryl-5-haloalkylpyrazoles and glyphosate, it's salts, diquat or paraquat MONSANTO COMPANY (US) 1996-07-16 US disclosed
US-5530126-A ALKYLATION IN INERT SOLVENT MONSANTO COMPANY (US) 1996-06-25 US disclosed
US-5496956-A BY ESTERIFICATION OF CARBOXY SUBSTITUTION WITH ALCOHOLS IN THE PRESENCE OF MINERAL ACID MONSANTO COMPANY (US) 1996-03-05 US disclosed
US-5489571-A CROP-SAFE COMPOUNDS EFFECTIVE AT LOW CONCENTRATIONS MONSANTO COMPANY (US) 1996-02-06 US disclosed
US-5281571-A Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles MONSANTO COMPANY (US) 1994-01-25 US disclosed
EP-0553307-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1993-08-04 EP disclosed
WO-1992006962-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1992-04-30 WO disclosed