SCHEMBL8565496

SCHEMBL8565496

CN1CCC(Nc2cc3c(Nc4ccc(F)c(Cl)c4)ncnc3cn2)CC1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.70
ERBB2 P04626 10/20 0.70
HPGD P15428 1/20 0.70
HTT P42858 1/20 0.70
ERBB4 Q15303 8/20 0.61
JAK3 P52333 2/20 0.61
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
GRM1 Q13255 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359359 0.93 EGFR (0.67) EGFRERBB2HPGDHTTERBB4
SCHEMBL8567653 0.87 EGFR (0.61) EGFRERBB2HPGDHTTERBB4
SCHEMBL8567648 0.87 EGFR (0.61) EGFRERBB2HPGDHTTERBB4
SCHEMBL7584450 0.85 ERBB2 (0.59) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL8569937 0.83 EGFR (0.62) EGFRERBB2HPGDHTTERBB4
SCHEMBL8567263 0.83 EGFR (0.61) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL8567268 0.83 EGFR (0.61) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL6904228 0.83 EGFR (0.61) EGFRERBB2HPGDHTT
Falnidamol SCHEMBL158563 0.82 EGFR (1.00) EGFRERBB2HPGDHTTERBB4
Falnidamol SCHEMBL29387986 0.82 EGFR (1.00) EGFRERBB2HPGDHTTERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885226-A1 4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997032881-A1 4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1997-09-12 WO disclosed