SCHEMBL8565644

SCHEMBL8565644

N#Cc1ccc2c(c1)CCC(N1CCC3(CC1)CC(O)c1cc4[nH]c(=O)[nH]c4cc1O3)C2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.68
HTR2A P28223 3/20 0.39
DRD2 P14416 2/20 0.39
KCNJ1 P48048 1/20 0.39
CYP11B2 P19099 1/20 0.37
ABCC9 O60706 2/20 0.34
ABCC8 Q09428 2/20 0.34
KCNJ11 Q14654 2/20 0.34
KCNJ8 Q15842 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
LMNA P02545 1/20 0.34
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
OPRL1 P41146 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570741 0.87 KCNH2 (0.53) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL8569350 0.85 KCNH2 (0.64) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL4706083 0.84 KCNH2 (0.74) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL8567782 0.84 KCNH2 (0.50) KCNH2HTR2ADRD2KCNJ1CYP11B2
Hydrochloric Acid SCHEMBL8564675 0.83 KCNH2 (0.49) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL8566025 0.82 KCNH2 (0.80) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL8831801 0.82 KCNH2 (0.72) KCNH2HTR2ADRD2KCNJ1CYP11B2
Hydrochloric Acid SCHEMBL8803788 0.81 KCNH2 (0.71) KCNH2HTR2ADRD2KCNJ1CYP11B2
Hydrochloric Acid SCHEMBL8832343 0.81 KCNH2 (0.71) KCNH2HTR2ADRD2KCNJ1CYP11B2
SCHEMBL8832003 0.81 KCNH2 (1.00) KCNH2HTR2ADRD2KCNJ1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP claimed
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed