SCHEMBL8565758

SCHEMBL8565758

Nc1ccc(CN2CCC3(CC2)CC(=O)c2cc(N)ccc2O3)cc1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.63
HDAC8 Q9BY41 9/20 0.59
HDAC6 Q9UBN7 9/20 0.59
HDAC3 O15379 8/20 0.59
HDAC4 P56524 8/20 0.59
HDAC1 Q13547 8/20 0.59
HDAC7 Q8WUI4 8/20 0.59
HDAC2 Q92769 8/20 0.59
HDAC10 Q969S8 8/20 0.59
HDAC11 Q96DB2 8/20 0.59
HDAC9 Q9UKV0 8/20 0.59
HDAC5 Q9UQL6 8/20 0.59
KCNH2 Q12809 2/20 0.55
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 1/20 0.45
FFAR1 O14842 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570725 0.85 HDAC3 (0.56) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL2506785 0.81 HDAC3 (0.57) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL4228161 0.80 SIGMAR1 (0.76) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL12017852 0.79 SIGMAR1 (0.74) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL1175467 0.79 SIGMAR1 (0.74) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL8565175 0.78 KCNH2 (0.71) HDAC8HDAC6HDAC3HDAC4HDAC1
SCHEMBL4270067 0.78 SIGMAR1 (1.00) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL8565539 0.77 KCNH2 (0.68) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL8185938 0.77 SIGMAR1 (0.84) SIGMAR1HDAC8HDAC6HDAC3HDAC4
SCHEMBL8184249 0.76 SIGMAR1 (0.82) SIGMAR1HDAC8HDAC6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed