SCHEMBL8566519

SCHEMBL8566519

CSC(=NC#N)NCc1ccc(CCO)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.36
CA2 P00918 1/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
CDK1 P06493 1/20 0.31
KDR P35968 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
SPHK1 Q9NYA1 1/20 0.31
EPHX2 P34913 1/20 0.30
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4679515 0.84 MEN1 (0.45) IDO1
SCHEMBL4679517 0.84 MEN1 (0.45) IDO1
SCHEMBL13325143 0.83 IDO1 (0.53) IDO1CA2
SCHEMBL19494294 0.83 IDO1 (0.53) IDO1CA2
SCHEMBL4886448 0.81 EPHX2 (0.49) EPHX2
SCHEMBL17731575 0.81 ALDH1A1 (0.50) TDP1EPHX2
SCHEMBL4886444 0.81 EPHX2 (0.49) EPHX2
SCHEMBL17731576 0.81 ALDH1A1 (0.50) TDP1EPHX2
SCHEMBL4685969 0.81 HTT (0.43)
SCHEMBL4685972 0.81 HTT (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed