SCHEMBL8566536

SCHEMBL8566536

COc1cc(-c2nn(C)c(C(F)(F)F)c2Br)c(F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.33
PDE2A O00408 1/20 0.33
GAA P10253 1/20 0.33
PPOX P50336 1/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HSP90AA1 P07900 2/20 0.32
HSP90AB1 P08238 2/20 0.32
CYP1A2 P05177 1/20 0.31
CCR1 P32246 2/20 0.31
BCAT2 O15382 1/20 0.31
BCAT1 P54687 1/20 0.31
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5398257 0.89 CYP1A2 (0.35) PDE10APDE2APPOXHTR2AHTR2C
SCHEMBL8549829 0.84 GAA (0.37) GAACYP1A2
SCHEMBL27814912 0.82 GAA (0.34) GAACYP1A2
SCHEMBL8570112 0.81 MAPT (0.34) GAACYP1A2
SCHEMBL14489535 0.79 PLAU (0.33) GAA
SCHEMBL3689455 0.79 RORC (0.36) GAA
SCHEMBL6912537 0.77 MEN1 (0.33) CYP1A2
SCHEMBL6911424 0.77 MEN1 (0.33) CYP1A2
SCHEMBL7609789 0.77 MEN1 (0.33) GAACYP1A2
SCHEMBL8566825 0.77 GAA (0.36) PDE10APDE2AGAAHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1050121-C Process for preparing substituted aryl-halogenoalkyl pyrazoles MONSANTO CO (US) 2000-03-08 CN disclosed
EP-0553307-B1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO CO (US) 1998-12-09 EP disclosed
EP-0791571-A1 Benzoyl derivatives MONSANTO COMPANY (US) 1997-08-27 EP disclosed
US-5536700-A Herbicidal compositions comprising aryl-5-haloalkylpyrazoles and glyphosate, it's salts, diquat or paraquat MONSANTO COMPANY (US) 1996-07-16 US disclosed
US-5530126-A ALKYLATION IN INERT SOLVENT MONSANTO COMPANY (US) 1996-06-25 US disclosed
US-5496956-A BY ESTERIFICATION OF CARBOXY SUBSTITUTION WITH ALCOHOLS IN THE PRESENCE OF MINERAL ACID MONSANTO COMPANY (US) 1996-03-05 US disclosed
US-5489571-A CROP-SAFE COMPOUNDS EFFECTIVE AT LOW CONCENTRATIONS MONSANTO COMPANY (US) 1996-02-06 US disclosed
US-5281571-A Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles MONSANTO COMPANY (US) 1994-01-25 US disclosed
EP-0553307-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1993-08-04 EP disclosed
WO-1992006962-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1992-04-30 WO disclosed