SCHEMBL8567008

SCHEMBL8567008

CS(=O)(=O)Nc1ccc2c(c1)C(=O)CC1(CCN(C3CCc4ccccc4C3)CC1)O2

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 4/20 0.55
KCNH2 Q12809 3/20 0.55
DRD2 P14416 1/20 0.51
HTR2A P28223 1/20 0.51
EPHX2 P34913 2/20 0.49
EPHX1 P07099 1/20 0.49
SCN5A Q14524 1/20 0.49
ADRA1A P35348 3/20 0.47
ADRA1B P35368 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8831700 0.99 ADRA1D (0.55) ADRA1DKCNH2DRD2HTR2AEPHX2
SCHEMBL8832305 0.95 KCNH2 (0.59) ADRA1DKCNH2DRD2HTR2AADRA1A
Hydrochloric Acid SCHEMBL8832204 0.94 KCNH2 (0.58) ADRA1DKCNH2DRD2HTR2AADRA1A
SCHEMBL8831650 0.91 KCNH2 (0.56) ADRA1DKCNH2DRD2HTR2AADRA1A
Hydrochloric Acid SCHEMBL8831670 0.91 KCNH2 (0.55) ADRA1DKCNH2DRD2HTR2AADRA1A
SCHEMBL7388074 0.88 KCNH2 (0.72) ADRA1DKCNH2HTR2AADRA1AADRA1B
SCHEMBL8831738 0.88 KCNH2 (0.72) ADRA1DKCNH2HTR2AADRA1AADRA1B
SCHEMBL8831813 0.88 KCNH2 (0.72) ADRA1DKCNH2HTR2AADRA1AADRA1B
SCHEMBL8831682 0.88 KCNH2 (0.55) ADRA1DKCNH2EPHX2EPHX1SCN5A
Hydrochloric Acid SCHEMBL8832193 0.88 KCNH2 (0.54) ADRA1DKCNH2EPHX2EPHX1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed