SCHEMBL8567015

SCHEMBL8567015

CC(C)(C)OC(=O)c1ccc(CCCOS(C)(=O)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CYP4A11 Q02928 3/20 0.43
CYP4F2 P78329 2/20 0.42
PPARG P37231 1/20 0.38
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MMP9 P14780 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
STAT3 P40763 2/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
MITF O75030 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720181 0.96 CA12 (0.45) CA1CA2CA12CA9CA14
SCHEMBL3126755 0.92 CA1 (0.48) CA1CA2CA12CA9CA14
SCHEMBL6488581 0.89 PLA2G4B (0.45) CA1CA2CA12CA9CA14
SCHEMBL6489468 0.85 PPARG (0.47) PPARG
SCHEMBL14415230 0.84 SLC7A5 (0.51) CA1CA2CA12CA9CA14
SCHEMBL3123864 0.84 CYP4A11 (0.62) CA1CA2CA12CA9CA14
SCHEMBL10984535 0.83 CA1 (0.38) CA1CA2CYP4A11CYP4F2PPARG
SCHEMBL23074190 0.82 CA2 (0.50) CA1CA2CA12CA9CA14
SCHEMBL6333378 0.82 HPGD (0.51) CA1CA2CA12CA9CA14
SCHEMBL9040138 0.81 RARB (0.53) CYP4A11CYP4F2KDM4EUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed