SCHEMBL8567258

SCHEMBL8567258

BrCCOc1ccc2nonc2c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.45
ENPP2 Q13822 2/20 0.41
NPC1 O15118 2/20 0.40
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 1/20 0.37
NCF1 P14598 8/20 0.36
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19122690 0.79 KMT2A (0.51) APPENPP2NPC1MAPTRAB9A
SCHEMBL9784162 0.78 HTR1B (0.47) NPC1MAPTRAB9APOLB
Bromide SCHEMBL9732194 0.77 HTR1B (0.46) NPC1MAPTRAB9APOLB
SCHEMBL7406721 0.72 APP (0.40) APPNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL17848625 0.72 APP (0.49) APPNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8146789 0.72 NPC1 (0.66) APPNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8363045 0.71 POLB (0.57) ENPP2NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8140756 0.71 NPC1 (0.47) NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL11016307 0.70 LTA4H (0.52) ENPP2NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL4017940 0.70 MAPT (0.44) APPENPP2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
US-5112824-A Benzofurazan compounds MERCK & CO., INC. (US) 1992-05-12 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed