SCHEMBL8567307

SCHEMBL8567307

CC1C(=O)c2cc(NS(C)(=O)=O)ccc2OC12CCN(CCc1ccc3nonc3c1)CC2

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.72
ADRA1D P25100 2/20 0.46
KCNJ1 P48048 3/20 0.44
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8570236 0.99 KCNH2 (0.71) KCNH2ADRA1DKCNJ1ADRA1A
SCHEMBL8563023 0.84 KCNH2 (1.00) KCNH2ADRA1DADRA1A
SCHEMBL8831725 0.84 KCNH2 (0.50) KCNH2ADRA1DADRA1A
SCHEMBL8561881 0.84 KCNH2 (0.50) KCNH2ADRA1DADRA1A
SCHEMBL8566922 0.83 KCNH2 (0.62) KCNH2ADRA1DKCNJ1
Hydrochloric Acid SCHEMBL8564930 0.83 KCNH2 (0.98) KCNH2ADRA1DADRA1A
Hydrochloric Acid SCHEMBL6375062 0.82 KCNH2 (0.97) KCNH2ADRA1DADRA1A
SCHEMBL8565294 0.80 ADRA1D (0.71) KCNH2ADRA1DADRA1A
SCHEMBL8564448 0.79 KCNH2 (0.75) KCNH2ADRA1DKCNJ1ADRA1A
Hydrochloric Acid SCHEMBL8569463 0.78 KCNH2 (0.78) KCNH2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP claimed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP claimed
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed