SCHEMBL8567340

SCHEMBL8567340

CC(C)C1=C[SiH](OCC[C@H](C)C[C@H](NC(=O)OC(C)(C)C)[C@@H](O)C[C@@H](C)C(=O)O)C(C(C)C)=C1C(C)C

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
KLK5 Q9Y337 1/20 0.34
APP P05067 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567921 0.74 CA1 (0.39) BACE1CA1CA2CA7BACE2
SCHEMBL8562900 0.74 CA1 (0.39) BACE1CA1CA2CA7BACE2
SCHEMBL5619596 0.67 KLK5 (0.62) BACE1KLK5APPPSEN1PSEN2
SCHEMBL9394616 0.67 KLK5 (0.62) BACE1KLK5APPPSEN1PSEN2
SCHEMBL6045015 0.64 KLK5 (0.41) BACE1KLK5
SCHEMBL6044435 0.64 KLK5 (0.45) BACE1KLK5APPPSEN1PSEN2
SCHEMBL6044566 0.64 REN (0.51) BACE1KLK5APPPSEN1PSEN2
SCHEMBL6044515 0.63 KLK5 (0.42) BACE1KLK5
SCHEMBL13413128 0.62 CA1 (0.53) BACE1CA1CA2CA7
SCHEMBL8562922 0.62 CYP2D6 (0.39) CA1CA2CA7KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed