SCHEMBL8567488

SCHEMBL8567488

C[C@]1(c2cc3ncccc3o2)CCCN1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.45
CHRNA4 P43681 2/20 0.45
ADAM17 P78536 2/20 0.35
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
PARP1 P09874 7/20 0.34
PARP2 Q9UGN5 3/20 0.34
TNKS O95271 1/20 0.34
PARP14 Q460N5 1/20 0.34
PARP10 Q53GL7 1/20 0.34
PARP12 Q9H0J9 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PARP4 Q9UKK3 1/20 0.34
PARP3 Q9Y6F1 1/20 0.34
PTGER3 P43115 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564031 0.78 CDC7 (0.32) PARP1PARP2TNKSPARP14PARP10
SCHEMBL8567997 0.78 CDC7 (0.32) PARP1PARP2TNKSPARP14PARP10
Hydrochloric Acid SCHEMBL8124451 0.78 PSMB5 (0.36) PARP1PARP2TNKSPARP14PARP10
SCHEMBL8565685 0.77 PARP1 (0.34) PARP1PARP2TNKSPARP14PARP10
SCHEMBL8114887 0.77 PARP1 (0.30) PARP1PARP2
SCHEMBL8570853 0.77 PARP1 (0.34) PARP1PARP2TNKSPARP14PARP10
SCHEMBL8120739 0.77 PARP1 (0.39) PARP1PARP2TNKSPARP14PARP10
SCHEMBL8128876 0.76 PTGER3 (0.32) PARP1PTGER3
SCHEMBL8121929 0.73 PARP1 (0.35) PARP1PARP2TNKSPARP14PARP10
Hydrochloric Acid SCHEMBL8120773 0.72 KDM4E (0.38) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842178-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1998-05-20 EP disclosed
WO-1997005139-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1997-02-13 WO disclosed