SCHEMBL8567650

SCHEMBL8567650

CCOc1cc(Cl)ccc1C(=O)N(C)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
TSHR P16473 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPT P10636 2/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
KCNMA1 Q12791 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP3A4 P08684 2/20 0.41
HPGD P15428 2/20 0.40
RAB9A P51151 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8571163 0.89 TSHR (0.49) TSHRMEN1KMT2AMAPTUSP2
SCHEMBL6333477 0.85 FLT1 (0.49) TSHRMEN1KMT2AMAPTRAB9A
SCHEMBL19840740 0.80 KDM4E (0.46) KDM4ETSHRMEN1KMT2ATDP1
SCHEMBL955961 0.80 CYP2C19 (0.49) KDM4EMEN1KMT2AMAPTUSP2
SCHEMBL305877 0.79 HCRTR1 (0.54) KDM4EMEN1KMT2AMAPTGAA
SCHEMBL7866445 0.79 TSHR (0.40) KDM4ETSHRMEN1KMT2AMAPT
SCHEMBL30628208 0.79 TSHR (0.61) KDM4ETSHRMEN1KMT2AMAPT
SCHEMBL1546386 0.79 TSHR (0.52) KDM4ETSHRMEN1KMT2AMAPT
SCHEMBL8444463 0.79 TSHR (0.61) KDM4ETSHRMEN1KMT2AMAPT
SCHEMBL3993311 0.79 KDM4E (0.49) KDM4ETSHRMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed