SCHEMBL19840740

SCHEMBL19840740

CCOc1cc(O[Si](C)(C)C)ccc1C(=O)N(C)OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
POLB P06746 2/20 0.38
HIF1A Q16665 1/20 0.37
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15782821 0.88 KMT2A (0.44) MEN1KMT2ATSHRCYP3A4CLK1
SCHEMBL8567650 0.80 KDM4E (0.42) KDM4EMEN1HPGDKMT2ASMN1; SMN2
SCHEMBL2647896 0.77 THRA (0.48) KDM4EALDH1A1MEN1KMT2APOLB
SCHEMBL955961 0.76 CYP2C19 (0.49) KDM4EALDH1A1HSD17B10MEN1HPGD
SCHEMBL305877 0.76 HCRTR1 (0.54) KDM4EALDH1A1HSD17B10MEN1HPGD
SCHEMBL4841763 0.74 NPC1 (0.57) ALDH1A1MEN1HPGDHTTKMT2A
SCHEMBL4097250 0.74 MAPT (0.50) ALDH1A1MEN1HTTKMT2ASMN1; SMN2
SCHEMBL25355846 0.73 KDM4E (0.43) KDM4EALDH1A1HSD17B10MEN1HPGD
SCHEMBL7866445 0.73 TSHR (0.40) KDM4EALDH1A1HSD17B10MEN1HPGD
SCHEMBL8045140 0.73 L3MBTL1 (0.39) KDM4EALDH1A1HSD17B10HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9884830-B2 Synthesis of tetracyclines and analogues thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2018-02-06 US disclosed