SCHEMBL8567807

SCHEMBL8567807

FC(F)(F)c1cccc(N2CCN(c3nc4ccccc4n4cccc34)CC2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.72
HTR1A P08908 6/20 0.72
TP53 P04637 2/20 0.70
MAPT P10636 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
HTR3E A5X5Y0 6/20 0.64
HTR3B O95264 6/20 0.64
HTR3A P46098 6/20 0.64
HTR3D Q70Z44 6/20 0.64
HTR3C Q8WXA8 6/20 0.64
HTR1D P28221 2/20 0.64
KDM4E B2RXH2 2/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2D6 P10635 1/20 0.64
TSHR P16473 1/20 0.64
NFKB1 P19838 1/20 0.64
CYP2C19 P33261 1/20 0.64
THPO P40225 1/20 0.64
HSD17B10 Q99714 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8880281 0.88 HTR2C (0.66) HTR2CHTR1ATP53MAPTSMN1; SMN2
SCHEMBL7298486 0.84 HTR2C (1.00) HTR2CHTR1ATP53MAPTSMN1; SMN2
SCHEMBL7296823 0.82 HTR2C (0.75) HTR2CHTR1ATP53MAPTSMN1; SMN2
SCHEMBL7296642 0.82 HTR2C (1.00) HTR2CHTR1ATP53MAPTSMN1; SMN2
SCHEMBL8567791 0.82 HTR3E (0.74) HTR2CHTR1AMAPTHTR3EHTR3B
SCHEMBL7298088 0.81 HTR2C (1.00) HTR2CHTR1ATP53MAPTSMN1; SMN2
SCHEMBL8566718 0.78 HTR3E (0.72) HTR2CHTR1ATP53MAPTHTR3E
SCHEMBL29390362 0.78 HTR3E (1.00) HTR2CHTR1ATP53HTR3EHTR3B
SCHEMBL1660466 0.78 HTR3E (1.00) HTR2CHTR1ATP53HTR3EHTR3B
SCHEMBL7298654 0.78 HTR2C (0.86) HTR2CHTR1ATP53MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed