SCHEMBL8568309

SCHEMBL8568309

Nc1nc(N)c2c(ccn2CCc2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)o2)n1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATIC P31939 14/20 0.53
SHMT1 P34896 13/20 0.53
SHMT2 P34897 13/20 0.53
GART P22102 10/20 0.52
FOLR2 P14207 1/20 0.47
FOLR1 P15328 1/20 0.47
DHFR P00374 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568317 1.00 ATIC (0.53) ATICSHMT1SHMT2GARTFOLR2
SCHEMBL8566866 0.95 ATIC (0.57) ATICSHMT1SHMT2GARTFOLR2
SCHEMBL8569542 0.87 ATIC (0.50) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8567736 0.86 ATIC (0.66) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8567743 0.86 ATIC (0.66) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571085 0.86 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571094 0.86 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001806 0.85 ATIC (0.72) ATICSHMT1SHMT2GARTFOLR2
SCHEMBL8562553 0.85 ATIC (0.48) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8562562 0.85 ATIC (0.48) ATICSHMT1SHMT2GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
CN-1070402-A The pyrimidine derivatives of condensation EISAI CO LTD (JP) 1993-03-31 CN disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed