SCHEMBL8568487

SCHEMBL8568487

CC[C@H](C)[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]2CCCN2C(=O)[C@H](C(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H]2CCCN2C1=O

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OXTR P30559 3/20 0.60
HDAC3 O15379 3/20 0.54
HDAC4 P56524 3/20 0.54
HDAC1 Q13547 3/20 0.54
HDAC7 Q8WUI4 3/20 0.54
HDAC2 Q92769 3/20 0.54
HDAC10 Q969S8 3/20 0.54
HDAC11 Q96DB2 3/20 0.54
HDAC8 Q9BY41 3/20 0.54
HDAC6 Q9UBN7 3/20 0.54
HDAC9 Q9UKV0 3/20 0.54
HDAC5 Q9UQL6 3/20 0.54
TACR1 P25103 3/20 0.52
TACR2 P21452 2/20 0.52
CIB1 Q99828 2/20 0.51
PDCD1 Q15116 1/20 0.50
CD274 Q9NZQ7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30179434 0.87 OXTR (0.68) OXTRHDAC3HDAC4HDAC1HDAC7
SCHEMBL31332253 0.86 HDAC3 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
Bq-123 SCHEMBL29388467 0.84 PDCD1 (0.60) OXTRHDAC3HDAC4HDAC1HDAC7
Bq-123 SCHEMBL11916897 0.84 PDCD1 (0.60) OXTRHDAC3HDAC4HDAC1HDAC7
Bq-123 SCHEMBL1290617 0.84 PDCD1 (0.60) OXTRHDAC3HDAC4HDAC1HDAC7
SCHEMBL16431734 0.82 HDAC3 (0.55) OXTRHDAC3HDAC4HDAC1HDAC7
SCHEMBL29553179 0.81 TACR1 (0.61) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24614245 0.81 HDAC3 (0.72) OXTRHDAC3HDAC4HDAC1HDAC7
SCHEMBL30833606 0.81 HDAC3 (0.72) OXTRHDAC3HDAC4HDAC1HDAC7
SCHEMBL19605615 0.81 HDAC3 (0.71) OXTRHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5801222-A Isolation and structure of the human cancer cell growth inhibitory cyclic octapeptides phakellistatin 10 and 11 ARIZONA BOARD OF REGENTS ACTING ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 1998-09-01 US claimed
US-5801222-A Isolation and structure of the human cancer cell growth inhibitory cyclic octapeptides phakellistatin 10 and 11 ARIZONA BOARD OF REGENTS ACTING ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 1998-09-01 US disclosed
US-5801222-A Isolation and structure of the human cancer cell growth inhibitory cyclic octapeptides phakellistatin 10 and 11 ARIZONA BOARD OF REGENTS ACTING ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 1998-09-01 US disclosed
US-5801222-A Isolation and structure of the human cancer cell growth inhibitory cyclic octapeptides phakellistatin 10 and 11 ARIZONA BOARD OF REGENTS ACTING ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 1998-09-01 US disclosed