SCHEMBL8569025

SCHEMBL8569025

CCCC=C(C#N)C(=O)OCC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.59
ALDH1A1 P00352 8/20 0.48
TSHR P16473 1/20 0.48
MAPT P10636 6/20 0.47
KDM4E B2RXH2 2/20 0.47
POLB P06746 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTP4A1 Q93096 1/20 0.47
MIF P14174 1/20 0.47
RAB9A P51151 5/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
NPC1 O15118 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
NPSR1 Q6W5P4 3/20 0.46
USP2 O75604 2/20 0.46
GAA P10253 2/20 0.46
LMNA P02545 1/20 0.46
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11256760 0.89 CYP2C9 (0.56) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL10899312 0.89 CYP2C9 (0.56) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL6696710 0.88 CYP2C9 (0.54) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL27741569 0.86 CYP2C9 (0.45) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL8053543 0.86 CYP2C9 (0.53) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL11208867 0.86 CYP2C9 (0.53) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL8600351 0.86 CYP2C9 (0.53) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL11269373 0.85 CYP2C9 (0.62) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL167038 0.85 CYP2C9 (0.62) CYP2C9ALDH1A1TSHRMAPTKDM4E
SCHEMBL7544282 0.84 ALDH1A1 (0.45) CYP2C9ALDH1A1TSHRMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843951-A Analgesic composition of pyrazolo(1,5-A) pyrimidines OTSUKA PHARMACEUTICAL FACTORY INC. (JP) 1998-12-01 US disclosed
EP-0795555-A1 ANALGESICS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1997-09-17 EP disclosed