SCHEMBL8569135

SCHEMBL8569135

COCC(=O)N(c1ccc(Cl)c(Cl)c1)C1CCNCC1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.72
TACR1 P25103 7/20 0.72
SLC6A2 P23975 9/20 0.45
SLC6A3 Q01959 8/20 0.45
KCNH2 Q12809 1/20 0.45
CHRM2 P08172 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL924943 0.86 SLC6A4 (0.67) SLC6A4TACR1SLC6A2SLC6A3KCNH2
SCHEMBL3035854 0.81 SLC6A4 (0.50) SLC6A4TACR1SLC6A2SLC6A3KCNH2
SCHEMBL8989455 0.81 TACR1 (0.49) SLC6A4TACR1SLC6A2SLC6A3KCNH2
Hydrochloric Acid SCHEMBL10977825 0.80 TACR1 (0.48) SLC6A4TACR1SLC6A2SLC6A3KCNH2
SCHEMBL8569723 0.79 CHRM2 (0.70) TACR1CHRM2CHRM3
SCHEMBL923866 0.79 TACR1 (0.55) SLC6A4TACR1SLC6A2SLC6A3KCNH2
SCHEMBL11571115 0.76 TACR1 (0.45) SLC6A4TACR1SLC6A3
Trifluoroacetic Acid SCHEMBL3029477 0.75 TACR1 (0.48) SLC6A4TACR1SLC6A2SLC6A3KCNH2
SCHEMBL8989462 0.74 TACR1 (0.46) SLC6A4TACR1SLC6A2SLC6A3
SCHEMBL926471 0.71 SLC6A4 (0.51) SLC6A4TACR1SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708101-B1 Piperidine derivatives, useful as neurokinin receptor antagonists ADIR (FR) 1998-12-09 EP disclosed
US-5652246-A NEUROKININ RECEPTOR ANTAGONISTS; NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-07-29 US disclosed
EP-0708101-A1 Novel piperidine derivatives, useful as neurokinin receptor antagonists ADIR ET COMPAGNIE (FR) 1996-04-24 EP disclosed