SCHEMBL8569334

SCHEMBL8569334

CC(C)(C)OC(=O)NC1CC2(C1)CN(Cc1ccccc1)C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
NPFFR1 Q9GZQ6 1/20 0.46
NPFFR2 Q9Y5X5 1/20 0.46
KCNA3 P22001 1/20 0.46
DRD2 P14416 4/20 0.44
KDM1A O60341 1/20 0.44
MAOB P27338 1/20 0.44
EPHX2 P34913 1/20 0.44
MEN1 O00255 2/20 0.43
CYP2D6 P10635 2/20 0.43
ALDH1A1 P00352 1/20 0.43
DRD4 P21917 1/20 0.42
ENPP2 Q13822 1/20 0.42
ATXN2 Q99700 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
JAK1 P23458 1/20 0.41
AKT1 P31749 1/20 0.41
DRD3 P35462 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14564141 0.89 KMT2A (0.54) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL6169636 0.87 KMT2A (0.55) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL1815532 0.84 KMT2A (0.65) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL23779786 0.83 KMT2A (0.55) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL6482327 0.83 KMT2A (0.55) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL18980315 0.83 KMT2A (0.55) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL20745275 0.82 KMT2A (0.54) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL27172319 0.82 ENPP2 (0.57) KMT2AL3MBTL1MEN1ALDH1A1ENPP2
SCHEMBL555251 0.81 KMT2A (0.62) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3
SCHEMBL17304781 0.81 KMT2A (0.65) KMT2AL3MBTL1NPFFR1NPFFR2KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230129359-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. 2023-04-27 US disclosed
US-20230129359-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. 2023-04-27 US disclosed
WO-2023010078-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2023-02-02 WO disclosed
WO-2021158698-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2021-08-12 WO disclosed
EP-0871628-A1 QUINOLIZINONE TYPE COMPOUNDS Abbott Laboratories (US) 1998-10-21 EP disclosed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230129359-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE CHRM4, CHRM2, CHRM5 KMT2A 1920/4885L3MBTL1 4078/4885NPFFR1 414/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.