SCHEMBL8569368

SCHEMBL8569368

Cc1c(N2CCC(C(=O)O)C2)c(F)cn2c(=O)c(C(=O)O)cc(C3CC3)c12

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.43
KCNH2 Q12809 5/20 0.41
NOTUM Q6P988 11/20 0.38
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8567049 0.99 SCN5A (0.43) SCN5AKCNH2NOTUMALDH1A1POLB
SCHEMBL7499390 0.91 SCN5A (0.45) SCN5AKCNH2ALDH1A1POLBCHRM2
SCHEMBL8569999 0.89 SCN5A (0.44) SCN5AKCNH2ALDH1A1POLBCHRM2
SCHEMBL5571872 0.89 SCN5A (0.44) SCN5AKCNH2ALDH1A1POLBCHRM2
SCHEMBL5571871 0.89 SCN5A (0.44) SCN5AKCNH2ALDH1A1POLBCHRM2
Abt-719 SCHEMBL1290190 0.88 ALDH1A1 (0.46) SCN5AKCNH2ALDH1A1POLBCHRM2
Abt-719 SCHEMBL1290350 0.88 ALDH1A1 (0.46) SCN5AKCNH2ALDH1A1POLBCHRM2
Hydrochloric Acid SCHEMBL7500623 0.88 SCN5A (0.43) SCN5AKCNH2ALDH1A1POLBCHRM2
Abt-719 SCHEMBL8569278 0.88 ALDH1A1 (0.46) SCN5AKCNH2ALDH1A1POLBCHRM2
SCHEMBL8563921 0.88 SCN5A (0.43) SCN5AKCNH2ALDH1A1POLBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US claimed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO claimed
EP-0871628-A1 QUINOLIZINONE TYPE COMPOUNDS Abbott Laboratories (US) 1998-10-21 EP disclosed
US-5726182-A TREATMENT OF BACTERIAL INFECTIONS ABBOTT LABORATORIES (US) 1998-03-10 US disclosed
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US disclosed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO disclosed