SCHEMBL8569458

SCHEMBL8569458

Cc1nc(N2CCc3ccccc3C2)nc(Cl)c1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.50
GRIN2D O15399 8/20 0.46
GRIN3B O60391 8/20 0.46
GRIN1 Q05586 8/20 0.46
GRIN2A Q12879 8/20 0.46
GRIN2B Q13224 8/20 0.46
GRIN2C Q14957 8/20 0.46
GRIN3A Q8TCU5 8/20 0.46
CHRM1 P11229 2/20 0.46
ADRA1D P25100 2/20 0.46
ADRA1A P35348 2/20 0.46
ADRA1B P35368 2/20 0.46
EED O75530 1/20 0.44
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572968 0.83 GRIN2D (0.46) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3682386 0.81 GRIN2D (0.56) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3714145 0.79 CETP (0.57) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6966650 0.77 CHRM3 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3676553 0.76 PTPN11 (0.47) CETPGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL6969378 0.76 GBA1 (0.49) CETPGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL8573962 0.76 GRIN2D (0.42) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8573444 0.75 GRIN2D (0.53) CETPGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL8573957 0.75 SMN1; SMN2 (0.44) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8572810 0.74 DRD1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1102144-C Noval pyrimidine derivatives and prepn. processes thereof YUHAN CORP (KR) 2003-02-26 CN disclosed
US-5750531-A ANTISECRETORY AGENTS FOR THE TREATMENT OF PEPTIC ULCER YUHAN CORPORATION (KR) 1998-05-12 US disclosed
CN-1155281-A Noval pyrimidine derivatives and prepn. processes thereof YUHAN CORP (KR) 1997-07-23 CN disclosed
EP-0775120-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 1997-05-28 EP disclosed
WO-1996005177-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1996-02-22 WO disclosed