SCHEMBL8569861

SCHEMBL8569861

Clc1cccc2c1ncc1cccn12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
KDM4E B2RXH2 7/20 0.54
HSD17B10 Q99714 3/20 0.54
GAA P10253 2/20 0.54
HPGD P15428 2/20 0.54
GLA P06280 1/20 0.54
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
RAB9A P51151 5/20 0.48
MAPK1 P28482 3/20 0.48
NPC1 O15118 3/20 0.48
MAPT P10636 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
ATM Q13315 1/20 0.48
CHEK1 O14757 1/20 0.39
LIMK1 P53667 1/20 0.39
MAPK14 Q16539 1/20 0.39
GFER P55789 1/20 0.38
PTPN1 P18031 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30963686 0.79 KDM4E (0.54) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL7401135 0.79 HAVCR2 (0.34) MEN1KMT2AMAPK14PTPN1PIM1
SCHEMBL2460831 0.77 FGFR1 (0.36) MEN1KMT2AGRM2HAVCR2LCK
SCHEMBL4146649 0.76 ALDH1A1 (0.51) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL7403844 0.75 ALDH1A1 (0.41) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL1079672 0.75 LCK (0.36) MAPK1GRM2HAVCR2SMN1; SMN2LCK
SCHEMBL1312899 0.74 KDM4E (0.49) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL8569567 0.73 KDM4E (0.47) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL8565559 0.72 DRD4 (0.45) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL29126966 0.72 ALDH1A1 (0.59) ALDH1A1KDM4EHSD17B10GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed