SCHEMBL8570296

SCHEMBL8570296

CCOC(=O)CCNCC#N

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.46
MGAM O43451 1/20 0.46
SI P14410 1/20 0.46
MGAM2 Q2M2H8 1/20 0.46
CYP1A2 P05177 1/20 0.42
LTA4H P09960 2/20 0.40
ALDH1A1 P00352 3/20 0.39
TRPA1 O75762 1/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.38
TOP2A P11388 1/20 0.38
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11188734 0.85 GAA (0.43) GAAMGAMSIMGAM2CYP1A2
SCHEMBL4464939 0.83 GAA (0.59) GAAMGAMSIMGAM2CYP1A2
SCHEMBL13756031 0.81 GAA (0.56) GAAMGAMSIMGAM2CYP1A2
Hydrochloric Acid SCHEMBL11851530 0.81 GAA (0.56) GAAMGAMSIMGAM2CYP1A2
SCHEMBL9774119 0.81 LTA4H (0.46) GAAMGAMSIMGAM2CYP1A2
SCHEMBL11343380 0.81 GAA (0.46) GAAMGAMSIMGAM2CYP1A2
SCHEMBL7434819 0.80 GAA (0.50) GAAMGAMSIMGAM2CYP1A2
SCHEMBL2969978 0.79 GAA (0.54) GAAMGAMSIMGAM2CYP1A2
SCHEMBL30893062 0.78 GAA (0.48) GAAMGAMSIMGAM2CYP1A2
SCHEMBL12939654 0.78 GAA (0.52) GAAMGAMSIMGAM2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed
US-4421693-A INSECTICIDES, MITICIDES OR NEMATOCIDES OTSUKA CHEMICAL CO., LTD. (JP) 1983-12-20 US disclosed
US-4413005-A 2,3-DIHYDRO-2,2-DIMETHYLBENZOFURAN-7-YL DERIVATIVES OTSUKA KAGAKU YAKUHIN KABUSHIKI KAISHA (JP) 1983-11-01 US disclosed